Humulus japonicus extract ameliorates collagen‑induced arthritis in mice through regulation of overall articular inflammation.

Humulus japonicus extract ameliorates collagen‑induced arthritis in mice through regulation of overall articular inflammation.

Humulus japonicus (HJ) is a widely used herbal remedy in Asia with anti-oxidative, anti-microbial and anti-inflammatory effects. We investigated the effect of HJ therapeutic potential in rheumatoid arthritis (RA) used a mouse model of collagen-induced arthritis (CIA) and lipopolysaccharide-stimulated murine macrophage cell line (RAW 264.7). CIA rats given 300 mg / kg orally HJ starting 3 days before the second immunization.

Clinical and histopathologic findings assessed in the rat paw CIA. Levels of autoantibodies and inflammatory markers are determined in plasma and cell culture supernatant, respectively. Expression at mRNA and protein levels were analyzed by quantitative reverse transcription-PCR and western blot analysis, respectively. HJ significantly decrease arthritic score dirty and foot swelling in CIA mice. Furthermore, synovial inflammation, cartilage damage and bone erosion that is markedly reduced by HJ.

It also decreased the expression of inflammatory enzymes in both paws of rats and RAW 264.7 cells. Moreover, the expression of genes associated with all pro-inflammatory macrophages and M1 macrophages significantly decreased, whereas the expression of anti-inflammatory M2 macrophage markers was significantly increased in the claws HJ-treated mice CIA. In addition, HJ reduced plasma levels of anti-type II collagen antibody following the decreased expression of T helper type 1 (Th1) and Th2-associated cell surface markers and cytokines in the claws.

HJ also significantly inhibited the expression of IL-6 both in vitro and in vivo, followed by a reduction in STAT3 phosphorylation and expression in rat paw CIA. Finally, the expression of genes associated with decreased osteoclast on HJ-treated rat paw CIA. These findings indicate that the HJ can play a role in suppressing the development of the CIA with the overall regulatory articular inflammation. These studies should provide new insights into the use of the HJ as a natural product effective therapy for RA.

Humulus japonicus extract ameliorates collagen‑induced arthritis in mice through regulation of overall articular inflammation.
Humulus japonicus extract ameliorates collagen‑induced arthritis in mice through regulation of overall articular inflammation.

Repeat-Dose Toxicity Studies AFPL1-Conjugate Vaccine Using Nicotine in male Sprague Dawley rats.

Tobacco smoking is the cause of 20% of deaths in Canada per year. Nicotine vaccine presents a promising alternative to traditional smoking cessation products, but until now, no vaccine has been able to move through all phases of clinical trials.

We have previously demonstrated that nicotine AFPL1-conjugate vaccine does not cause systemic or immunotoxicity in this mouse model and that heterologous vaccination approach is more profitable than these homologous to stimulate mucosal and systemic antibody anti-nicotine.

The purpose of this study was to confirm the safety profile of the vaccine in the repeated-dose toxicity studies. Heterologous vaccination strategy re-used, and Sprague-Dawley rats given a dose five times greater than in our previous studies.

Goat Anti Mouse IgA Polyclonal Affinity Purified

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Rabbit anti-Mouse Moesin IgG, affinity purified

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Anti-Per.C6Ð’ Affinity Purified HRP, Goat

PC118AF-HRP 1 mg
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VC807-AFB 1 mg
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Glutathione-S-transferase (GST) Affinity Purified Antibody

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Mouse Monoclonal Anti-Human IgM, clone 1, Affinity Purified (Bulk)

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Cy5 Conjugated Affinity Purified anti-Mouse IgG [H&L] [Goat]

SC012 250 µg
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EUR 81
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IRBAT7TAP100UG each
EUR 404
Description: Rabbit Anti T7 Tag Polyclonal Affinity Purified

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IRBAT7TAP1MG each
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Description: Rabbit Anti T7 Tag Polyclonal Affinity Purified

Cy2 Conjugated Affinity Purified anti-Mouse IgG [H&L] [Donkey]

SC011 250 µg
EUR 145

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IRBASTAGAP100UG each
EUR 404
Description: Rabbit Anti S-Tag Polyclonal Affinity Purified

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IRBASTAGAP1MG each
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Description: Rabbit Anti S-Tag Polyclonal Affinity Purified

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IRBAAU1TAP100UG each
EUR 404
Description: Rabbit Anti AU1 Tag Polyclonal Affinity Purified

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EUR 1550
Description: Rabbit Anti AU1 Tag Polyclonal Affinity Purified

Rabbit Anti GST Tag Polyclonal Affinity Purified

IRBAGSTTAP100UG each
EUR 184
Description: Rabbit Anti GST Tag Polyclonal Affinity Purified

Rabbit Anti GST Tag Polyclonal Affinity Purified

IRBAGSTTAP1MG each
EUR 919
Description: Rabbit Anti GST Tag Polyclonal Affinity Purified

Rabbit Anti HSV Tag Polyclonal Affinity Purified

IRBAHSVTAP100UG each
EUR 404
Description: Rabbit Anti HSV Tag Polyclonal Affinity Purified

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IRBAHSVTAP1MG each
EUR 1550
Description: Rabbit Anti HSV Tag Polyclonal Affinity Purified

Goat Anti Horse IgM Polyclonal Affinity Purified

IGTAHSIGMAP1MG each
EUR 161
Description: Goat Anti Horse IgM Polyclonal Affinity Purified

Goat Anti Human IgA Polyclonal Affinity Purified

IGTAHUIGAAP1MG each
EUR 143
Description: Goat Anti Human IgA Polyclonal Affinity Purified

Goat Anti Human IgE Polyclonal Affinity Purified

IGTAHUIGEAP1MG each
EUR 252
Description: Goat Anti Human IgE Polyclonal Affinity Purified

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IGTAHUIGGAP1MG each
EUR 111
Description: Goat Anti Human IgG Polyclonal Affinity Purified

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IGTAHUIGMAP1MG each
EUR 155
Description: Goat Anti Human IgM Polyclonal Affinity Purified

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IGTAHUIGMAP500UG each
EUR 103
Description: Goat Anti Human IgM Polyclonal Affinity Purified

Goat Anti Llama IgG Polyclonal Affinity Purified

IGTALLIGGAP1000MG each
EUR 5325
Description: Goat Anti Llama IgG Polyclonal Affinity Purified

Goat Anti Llama IgG Polyclonal Affinity Purified

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EUR 1067
Description: Goat Anti Llama IgG Polyclonal Affinity Purified

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IGTALLIGGAP10MG each
EUR 172
Description: Goat Anti Llama IgG Polyclonal Affinity Purified

Chicken Anti HA Tag Polyclonal Affinity Purified

ICHAHATAP100UG each
EUR 404
Description: Chicken Anti HA Tag Polyclonal Affinity Purified

Chicken Anti HA Tag Polyclonal Affinity Purified

ICHAHATAP1MG each
EUR 1550
Description: Chicken Anti HA Tag Polyclonal Affinity Purified

Anti-SF9 Insect Cell HCP 2G affinity purified

SF9RB01-AF 0.5 mg
EUR 2295.6
Description: Anti-SF9 Insect Cell HCP 2G affinity purified by Cygnus Technologies is available in Europe via Gentaur.

Rabbit Anti Rat ACE2 Polyclonal Affinity Purified

IRBARTACE2AP100UG each
EUR 509
Description: Rabbit Anti Rat ACE2 Polyclonal Affinity Purified

*Sheep Anti Human tPA Polyclonal Affinity Purified

ISHAHUTPAAP100UG each
EUR 533
Description: *Sheep Anti Human tPA Polyclonal Affinity Purified

Rabbit Anti Goat IgG Polyclonal Affinity Purified

IRBAGTIGGAP1MG each
EUR 143
Description: Rabbit Anti Goat IgG Polyclonal Affinity Purified

Goat Anti Bovine IgG Polyclonal Affinity Purified

IGTABOIGGAP1MG each
EUR 192
Description: Goat Anti Bovine IgG Polyclonal Affinity Purified

Goat Anti Canine IgA Polyclonal Affinity Purified

IGTACNIGAAP1MG each
EUR 242
Description: Goat Anti Canine IgA Polyclonal Affinity Purified

Goat Anti Canine IgE Polyclonal Affinity Purified

IGTACNIGEAP1MG each
EUR 624
Description: Goat Anti Canine IgE Polyclonal Affinity Purified

Goat Anti Canine IgG Polyclonal Affinity Purified

IGTACNIGGAP1MG each
EUR 221
Description: Goat Anti Canine IgG Polyclonal Affinity Purified

Goat Anti Feline IgA Polyclonal Affinity Purified

IGTAFEIGAAP1MG each
EUR 154
Description: Goat Anti Feline IgA Polyclonal Affinity Purified

Goat Anti Feline IgG Polyclonal Affinity Purified

IGTAFEIGGAP1MG each
EUR 143
Description: Goat Anti Feline IgG Polyclonal Affinity Purified

Goat Anti Feline IgM Polyclonal Affinity Purified

IGTAFEIGMAP1MG each
EUR 220
Description: Goat Anti Feline IgM Polyclonal Affinity Purified

Goat Anti Rabbit IgG Polyclonal Affinity Purified

IGTARBIGGAP1MG each
EUR 111
Description: Goat Anti Rabbit IgG Polyclonal Affinity Purified

Goat Anti Rabbit IgM Polyclonal Affinity Purified

IGTARBIGMAP1MG each
EUR 185
Description: Goat Anti Rabbit IgM Polyclonal Affinity Purified

*Mouse IgG Affinity Purified Endotoxin Depleted

IMSIGGAPLX50MG each
EUR 503
Description: *Mouse IgG Affinity Purified Endotoxin Depleted

Rabbit Anti Sheep IgG Polyclonal Affinity Purified

IRBASHIGGAP1MG each
EUR 143
Description: Rabbit Anti Sheep IgG Polyclonal Affinity Purified

Goat Anti Chicken IgA Polyclonal Affinity Purified

IGTACHIGAAP1MG each
EUR 235
Description: Goat Anti Chicken IgA Polyclonal Affinity Purified

Goat Anti Chicken IgY Polyclonal Affinity Purified

IGTACHIGYAP1MG each
EUR 132
Description: Goat Anti Chicken IgY Polyclonal Affinity Purified

Goat Anti Hamster IgG Polyclonal Affinity Purified

IGTAHMIGGAP1MG each
EUR 145
Description: Goat Anti Hamster IgG Polyclonal Affinity Purified

Goat Anti Hamster IgG Polyclonal Affinity Purified

IGTAHMIGGAP500UG each
EUR 156
Description: Goat Anti Hamster IgG Polyclonal Affinity Purified

*Rabbit Anti Human tPA Polyclonal Affinity Purified

IRBAHUTPAAP100UG each
EUR 481
Description: *Rabbit Anti Human tPA Polyclonal Affinity Purified

*Rabbit Anti Human tPA Polyclonal Affinity Purified

IRBAHUTPAAP1MG each
EUR 3891
Description: *Rabbit Anti Human tPA Polyclonal Affinity Purified

Rabbit Anti Llama IgG Polyclonal Affinity Purified

IRBALLIGGAP1000MG each
EUR 7454
Description: Rabbit Anti Llama IgG Polyclonal Affinity Purified

Rabbit Anti Llama IgG Polyclonal Affinity Purified

IRBALLIGGAP100MG each
EUR 1918
Description: Rabbit Anti Llama IgG Polyclonal Affinity Purified

Rabbit Anti Llama IgG Polyclonal Affinity Purified

IRBALLIGGAP10MG each
EUR 258
Description: Rabbit Anti Llama IgG Polyclonal Affinity Purified

Rabbit Anti Human IgG Polyclonal Affinity Purified

IRBAHUIGGAP1MG each
EUR 143
Description: Rabbit Anti Human IgG Polyclonal Affinity Purified

physiological conditions, food and water consumption, body temperature, inflammation of the injection site, relative organ weights, histopathology, and blood chemistry and hematology were evaluated during the vaccination period to determine the safety of the vaccine. AFPL1 nicotine-conjugate vaccine does not induce clinically relevant changes or induces symptoms that would be associated with toxicity, making it a promising candidate for future investigations.

Nathaniel

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